SCHEMBL22703621

SCHEMBL22703621

COC(=O)C1CCN(CCCNC(=O)OC(C)(C)C)CC1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.54
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 1/20 0.48
TSHR P16473 1/20 0.48
SIGMAR1 Q99720 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
CACNA1H O95180 1/20 0.44
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
EPHX1 P07099 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22470192 0.92 DRD2 (0.52) DRD2MEN1KMT2AALDH1A1TSHR
SCHEMBL22699069 0.85 DRD2 (0.54) DRD2MEN1KMT2ASIGMAR1TDP1
SCHEMBL18947871 0.85 DRD2 (0.54) DRD2MEN1KMT2ASIGMAR1TDP1
SCHEMBL24619896 0.85 DRD2 (0.54) DRD2MEN1KMT2ASIGMAR1TDP1
SCHEMBL31687516 0.85 ACKR3 (0.53) DRD2MEN1KMT2ASIGMAR1TDP1
SCHEMBL8254760 0.84 DRD2 (0.64) DRD2MEN1KMT2AALDH1A1SIGMAR1
SCHEMBL32690155 0.84 DRD2 (0.47) DRD2MEN1KMT2AALDH1A1TSHR
SCHEMBL6700 0.84 DRD2 (0.53) DRD2MEN1KMT2ASIGMAR1TDP1
SCHEMBL21815267 0.83 DRD2 (0.50) DRD2MEN1KMT2ASIGMAR1TDP1
SCHEMBL9281583 0.82 SMN1; SMN2 (0.50) MEN1KMT2AALDH1A1TSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020236690-A1 NATRIURETIC PEPTIDE RECEPTOR A AGONISTS USEFUL FOR THE TREATMENT OF CARDIOMETABOLIC DISEASES, KIDNEY DISEASE AND DIABETES MERCK SHARP & DOHME CORP. (US) 2020-11-26 WO disclosed