SCHEMBL22709347

SCHEMBL22709347

COC(=O)CC1(CCCC(=O)O)CCc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC9 Q9UKV0 1/20 0.38
OPRL1 P41146 1/20 0.37
TACR1 P25103 1/20 0.37
TACR3 P29371 1/20 0.37
TSHR P16473 1/20 0.36
KDM1A O60341 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR2C P28335 1/20 0.36
SLC6A3 Q01959 1/20 0.36
NOTUM Q6P988 1/20 0.36
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22709565 0.93 ALDH1A1 (0.40) HDAC9ALDH1A1
SCHEMBL22709350 0.93 NOTUM (0.40) HDAC9OPRL1TACR1TACR3NOTUM
SCHEMBL24483073 0.87 NOTUM (0.41) HDAC9TACR1TACR3NOTUM
SCHEMBL22709563 0.85 KMT2A (0.39) KDM1ANOTUM
SCHEMBL22692094 0.85 DGAT1 (0.44) HTR2C
SCHEMBL22692045 0.85 DGAT1 (0.44) HTR2C
SCHEMBL22692046 0.85 DGAT1 (0.44) HTR2C
SCHEMBL30067249 0.84 CHRNA7 (0.35) HDAC9OPRL1TACR1TACR3
SCHEMBL22709344 0.83 ALDH1A1 (0.37) HDAC9OPRL1TACR1TACR3ALDH1A1
SCHEMBL24483072 0.81 SIGMAR1 (0.36) HDAC9TACR1TACR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022115439-A1 KRAS G12C INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-06-02 WO disclosed
WO-2020236940-A1 KRAS G12C INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2020-11-26 WO disclosed