SCHEMBL22717364

SCHEMBL22717364

C[Si](C)(C)CCOCn1ccc(C(O)c2ccccc2)n1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.31
F2RL1 P55085 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
F11 P03951 1/20 0.31
LTA4H P09960 1/20 0.30
ALDH1A1 P00352 2/20 0.30
HTT P42858 1/20 0.30
CYP19A1 P11511 2/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31283459 0.82 F2RL1 (0.31) NPC1F2RL1
SCHEMBL13326840 0.80
SCHEMBL31056357 0.78 DGAT1 (0.33)
SCHEMBL31708798 0.78 F2RL1 (0.32) F2RL1
SCHEMBL24102105 0.77 NPC1 (0.31) NPC1
SCHEMBL31283365 0.76 DGAT1 (0.30)
SCHEMBL26453175 0.74 KMT2A (0.45) KDM4ENPC1NPSR1ALDH1A1CYP19A1
SCHEMBL17049033 0.74 ALDH1A1 (0.33) KDM4EALDH1A1MAPT
SCHEMBL26910784 0.74
SCHEMBL19926702 0.72 NPC1 (0.33) NPC1F11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3976618-A1 TRICYCLIC COMPOUNDS Aligos Therapeutics, Inc. (US) 2022-04-06 EP disclosed
US-20220000874-A1 TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. 2022-01-06 US disclosed
US-20220000874-A1 TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. 2022-01-06 US disclosed
US-11136321-B2 Tricyclic compounds ALIGOS THERAPEUTICS, INC. (US) 2021-10-05 US disclosed
US-11136321-B2 Tricyclic compounds ALIGOS THERAPEUTICS, INC. (US) 2021-10-05 US disclosed
US-20200407361-A1 TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. 2020-12-31 US disclosed
US-20200407361-A1 TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. 2020-12-31 US disclosed
WO-2020243199-A1 TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. (US) 2020-12-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220000874-A1 TRICYCLIC COMPOUNDS SLC10A1, PKD1, CEL KDM4E 4358/4885NPC1 5/4885TSHR 2105/4885
US-11136321-B2 Tricyclic compounds SLC10A1, PKD1, CEL KDM4E 4358/4885NPC1 5/4885TSHR 2105/4885
US-20200407361-A1 TRICYCLIC COMPOUNDS SLC10A1, PKD1, CEL KDM4E 4358/4885NPC1 5/4885TSHR 2105/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.