SCHEMBL22720267

SCHEMBL22720267

COc1nc(C=Cc2c(F)cccc2OC)c(CN(C)C(=O)OC(C)(C)C)c(N2CCN(C(=O)O)C(C(C)(C)C)C2)n1

nearest known ligand 0.31

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.31
SLC6A4 P31645 2/20 0.31
HTR2A P28223 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
LIMK2 P53671 1/20 0.31
RAB9A P51151 1/20 0.30
NPY2R P49146 1/20 0.30
TLR9 Q9NR96 1/20 0.30
TLR7 Q9NYK1 1/20 0.30
FFAR2 O15552 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28530744 0.89 TLR9 (0.35) HTR2CSLC6A4HTR2AALDH1A1SMN1; SMN2
SCHEMBL28544155 0.89 TLR9 (0.35) HTR2CSLC6A4HTR2AALDH1A1SMN1; SMN2
SCHEMBL22720265 0.85 TLR9 (0.40) TLR9TLR7
SCHEMBL22724634 0.76 KRAS (0.39) HTR2CSLC6A4HTR2ATLR9TLR7
SCHEMBL22720270 0.69 KRAS (0.37)
SCHEMBL28537273 0.67 TLR9 (0.35) HTR2CSLC6A4TLR9TLR7
SCHEMBL18128721 0.64 KRAS (0.38) LIMK2
SCHEMBL2760636 0.64 DRD2 (0.51) ALDH1A1SMN1; SMN2
SCHEMBL18128367 0.63 KRAS (0.36) ALDH1A1LIMK2
SCHEMBL12454614 0.62 RIPK1 (0.46) HTR2CSLC6A4HTR2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed