SCHEMBL28537273

SCHEMBL28537273

COc1nc(C)c(CN(C)C(=O)OC(C)(C)C)c(N2CCN(C(=O)O)CC2)n1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 3/20 0.35
TLR7 Q9NYK1 2/20 0.34
HTR2C P28335 1/20 0.31
SLC6A4 P31645 1/20 0.31
GBA1 P04062 1/20 0.30
CACNA1G O43497 1/20 0.30
CACNA1B Q00975 1/20 0.30
CACNA1C Q13936 1/20 0.30
SMPD3 Q9NY59 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720279 0.92 TLR9 (0.43) TLR9TLR7GBA1SMPD3
SCHEMBL28542868 0.82 KRAS (0.39)
SCHEMBL28542866 0.82 KRAS (0.39)
SCHEMBL29127300 0.82 TLR9 (0.35) TLR9TLR7HTR2CSLC6A4CACNA1G
SCHEMBL28530744 0.77 TLR9 (0.35) TLR9TLR7HTR2CSLC6A4
SCHEMBL28544155 0.77 TLR9 (0.35) TLR9TLR7HTR2CSLC6A4
SCHEMBL22720268 0.75 KRAS (0.39) TLR9
SCHEMBL22720270 0.72 KRAS (0.37)
SCHEMBL22720265 0.70 TLR9 (0.40) TLR9TLR7
SCHEMBL22720236 0.69 TLR9 (0.44) TLR9TLR7GBA1SMPD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396147-A Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-14 CN disclosed
CN-112552294-A Piperazine heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-03-26 CN disclosed