SCHEMBL22720265

SCHEMBL22720265

COc1nc(/C=C/c2c(F)cccc2OC)c(CN(C)C(=O)OC(C)(C)C)c(N2CCN(C(=O)OC(C)(C)C)CC2)n1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 5/20 0.40
TLR7 Q9NYK1 2/20 0.40
CXCR2 P25025 1/20 0.40
ABCB1 P08183 2/20 0.35
ALK Q9UM73 1/20 0.35
GPR119 Q8TDV5 2/20 0.35
DNMT3A Q9Y6K1 1/20 0.35
RORC P51449 1/20 0.35
KDM1A O60341 1/20 0.34
GALR2 O43603 1/20 0.34
GALR1 P47211 1/20 0.34
ACHE P22303 1/20 0.34
TGFBR1 P36897 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28544155 0.94 TLR9 (0.35) TLR9TLR7CXCR2TP53
SCHEMBL28530744 0.94 TLR9 (0.35) TLR9TLR7CXCR2TP53
SCHEMBL22724634 0.89 KRAS (0.39) TLR9TLR7CXCR2
SCHEMBL22720267 0.85 HTR2C (0.31) TLR9TLR7
SCHEMBL22720279 0.77 TLR9 (0.43) TLR9TLR7GPR119ACHE
SCHEMBL28537273 0.70 TLR9 (0.35) TLR9TLR7
SCHEMBL31651847 0.68 ALDH1A1 (0.45) ABCB1ALKGPR119TP53
SCHEMBL23119215 0.67 GRM5 (0.45) ABCB1GPR119TGFBR1
SCHEMBL12454614 0.65 RIPK1 (0.46)
SCHEMBL22720268 0.65 KRAS (0.39) TLR9GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed