SCHEMBL22720279

SCHEMBL22720279

COc1nc(C)c(CN(C)C(=O)OC(C)(C)C)c(N2CCN(C(=O)OC(C)(C)C)CC2)n1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 3/20 0.43
TLR7 Q9NYK1 2/20 0.39
SMPD3 Q9NY59 1/20 0.37
TLR8 Q9NR97 1/20 0.36
DPP4 P27487 1/20 0.36
GPR119 Q8TDV5 5/20 0.36
GBA1 P04062 2/20 0.36
CKS1B P61024 1/20 0.35
SKP1 P63208 1/20 0.35
SKP2 Q13309 1/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ACHE P22303 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAP4K4 O95819 1/20 0.34
KIT P10721 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720268 0.82 KRAS (0.39) TLR9GPR119
SCHEMBL22724587 0.78 TLR9 (0.44) TLR9TLR7SMPD3GBA1CKS1B
SCHEMBL22720236 0.78 TLR9 (0.44) TLR9TLR7SMPD3GBA1CKS1B
SCHEMBL22720265 0.77 TLR9 (0.40) TLR9TLR7GPR119ACHE
SCHEMBL22720228 0.76 TLR9 (0.42) TLR9TLR7SMPD3GPR119GBA1
SCHEMBL21734104 0.70 GBA1 (0.44) TLR9GPR119GBA1CKS1BSKP1
SCHEMBL19636828 0.69 TLR9 (0.40) TLR9TLR7GPR119GBA1CKS1B
SCHEMBL22873609 0.68 GPR119 (0.55) TLR9SMPD3GPR119GBA1CKS1B
SCHEMBL31652099 0.68 TLR9 (0.54) TLR9TLR7SMPD3GPR119GBA1
SCHEMBL5851554 0.67 P2RY12 (0.48) TLR9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed