SCHEMBL22723932

SCHEMBL22723932

CCN1CCc2ccc(CC(C)C)nc2CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
DRD2 P14416 3/20 0.37
DRD1 P21728 2/20 0.37
LMNA P02545 4/20 0.36
PNMT P11086 1/20 0.36
RAD52 P43351 1/20 0.36
RECQL P46063 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
KCNH2 Q12809 1/20 0.36
GRM5 P41594 2/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.34
HSP90AB1 P08238 1/20 0.34
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22723975 0.79 DRD3 (0.35) CYP3A4TSHRHSD17B10DRD2DRD1
SCHEMBL11639939 0.78 ADRA2A (0.40) TSHRALDH1A1
SCHEMBL22387665 0.78 ADRA2A (0.37) TSHRRXFP1
SCHEMBL24253486 0.78 MAOA (0.40) DRD2DRD1DRD4DRD5HRH3
SCHEMBL22993267 0.78 CYP2C19 (0.43) TSHRHSD17B10RECQLKCNH2ALDH1A1
SCHEMBL21730188 0.77 MAPT (0.36) GRM5MAPTHRH3
SCHEMBL28890009 0.72 MAPT (0.40) LMNAPNMTRAD52RECQLGRM5
SCHEMBL24221619 0.71 GRM5 (0.32) GRM5
SCHEMBL24221623 0.71 GRM5 (0.33) TSHRHSD17B10DRD2DRD1LMNA
SCHEMBL22723964 0.70 DRD3 (0.51) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3744721-A1 CONDENSED CYCLIC COMPOUND HAVING DOPAMINE D3 RECEPTOR ANTAGONISM Shionogi & Co., Ltd (JP) 2020-12-02 EP disclosed