SCHEMBL22744121

SCHEMBL22744121

C#C[C@H](O)c1ncccn1

nearest known ligand 0.30

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
PKM P14618 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
ATM Q13315 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3758698 0.73 SLC6A2 (0.45) ALDH1A1MAPTPKMHPGDHTT
SCHEMBL30321098 0.73 SLC6A2 (0.45) ALDH1A1MAPTPKMHPGDHTT
SCHEMBL22744059 0.73 SLC6A2 (0.45) ALDH1A1MAPTPKMHPGDHTT
SCHEMBL22744134 0.70 HDAC8 (0.34) HDAC8
SCHEMBL3082231 0.69
SCHEMBL22031546 0.69 NAPRT (0.39) L3MBTL1
SCHEMBL17681988 0.69 P2RX7 (0.35)
SCHEMBL17682018 0.69 P2RX7 (0.35)
SCHEMBL8765939 0.69 CES2 (0.34) ALDH1A1MAPTHTTNPSR1L3MBTL1
SCHEMBL31570465 0.66 TRPM8 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239999-A1 SMALL MOLECULE INHIBITORS OF NF-kB INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2020-12-03 WO disclosed