SCHEMBL8765939

SCHEMBL8765939

C#CC(C(=O)O)c1ncccn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
PTPRA P18433 1/20 0.34
NAPRT Q6XQN6 3/20 0.33
LMNA P02545 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
P4HTM Q9NXG6 1/20 0.33
KDM4E B2RXH2 5/20 0.32
TDP1 Q9NUW8 2/20 0.32
ALDH1A1 P00352 2/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
BLM P54132 1/20 0.31
AGER Q15109 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CYP1A2 P05177 1/20 0.31
GAA P10253 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8831554 0.71 PTGS2 (0.42) PTPRANAPRTLMNAL3MBTL1P4HTM
SCHEMBL6999564 0.70 SRC (0.44) CES2CES1PTPRANAPRTLMNA
Hydrochloric Acid SCHEMBL22775404 0.70 PTGS2 (0.41) PTPRANAPRTLMNAL3MBTL1P4HTM
SCHEMBL7527146 0.70 SRC (0.50) CES2CES1LMNAL3MBTL1KDM4E
SCHEMBL8766788 0.69 KDM4E (0.41) NAPRTLMNAKDM4ETSHRGAA
SCHEMBL22744121 0.69 HDAC8 (0.30) L3MBTL1ALDH1A1MAPTNPSR1HTT
SCHEMBL8766512 0.68 CYP1A2 (0.41) CES1NAPRTALDH1A1CYP1A2
SCHEMBL86412 0.65 MEN1 (0.44) LMNAL3MBTL1ALDH1A1CYP1A2GAA
SCHEMBL22744134 0.64 HDAC8 (0.34)
SCHEMBL24327756 0.62 KMT2A (0.35) PTPRANAPRTLMNAL3MBTL1P4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1997-07-30 EP disclosed
WO-1996011686-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-04-25 WO disclosed