SCHEMBL22760046

SCHEMBL22760046

O=C(O)c1c(N2CCCCC2)c2cc(Cl)c(Br)cc2n1-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.38
ALDH1A1 P00352 4/20 0.36
HPGD P15428 3/20 0.36
HSD17B10 Q99714 3/20 0.36
GAA P10253 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALOX15 P16050 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAPT P10636 2/20 0.36
TSHR P16473 2/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
EDNRA P25101 1/20 0.36
LMNA P02545 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760357 0.95 REN (0.38) RENALDH1A1HPGDHSD17B10GAA
SCHEMBL22747915 0.91 ALDH1A1 (0.40) RENALDH1A1HPGDHSD17B10GAA
SCHEMBL22747873 0.89 MAT2A (0.43) ALDH1A1HPGDGAAMEN1KMT2A
SCHEMBL22760176 0.86 REN (0.38) RENALDH1A1HPGDHSD17B10GAA
SCHEMBL22760356 0.84 MAT2A (0.43) ALDH1A1HPGDGAAMEN1KMT2A
SCHEMBL22747827 0.83 SMN1; SMN2 (0.42) ALDH1A1HPGDHSD17B10GAAMEN1
SCHEMBL22748254 0.82 MAT2A (0.46) RENEDNRAFABP3FABP4FABP5
SCHEMBL22760383 0.82 GAA (0.32) RENALDH1A1HPGDHSD17B10GAA
SCHEMBL22748265 0.81 HPGD (0.40) RENALDH1A1HPGDHSD17B10GAA
SCHEMBL22760058 0.81 ALDH1A1 (0.39) ALDH1A1HPGDGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed