SCHEMBL22760116

SCHEMBL22760116

CCOC(=O)c1c(N2CCCCC2)c2c(Cl)cc(Cl)cc2n1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 2/20 0.47
HPGD P15428 3/20 0.43
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
LMNA P02545 1/20 0.40
MAPK1 P28482 1/20 0.40
KDM4E B2RXH2 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
TP53 P04637 1/20 0.39
MAT2A P31153 1/20 0.39
HIF1A Q16665 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
DYRK1A Q13627 1/20 0.39
TSHR P16473 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760184 0.86 MAPK8 (0.48) ALDH1A1MAPTGAAHPGDMAT2A
SCHEMBL22760086 0.85 MAT2A (0.43) ALDH1A1MAPTGAAHPGDMEN1
SCHEMBL22760115 0.84 MAPT (0.46) ALDH1A1MAPTGAAHPGDMEN1
SCHEMBL22760359 0.82 ALDH1A1 (0.46) ALDH1A1MAPTGAAHPGDMEN1
SCHEMBL22760172 0.82 MAPT (0.47) ALDH1A1MAPTGAAHPGDMEN1
SCHEMBL22747837 0.81 ALDH1A1 (0.45) ALDH1A1MAPTGAAHPGDMEN1
SCHEMBL22747885 0.79 HPGD (0.45) ALDH1A1MAPTGAAHPGDMEN1
SCHEMBL22760215 0.79 HPGD (0.51) ALDH1A1MAPTGAAHPGDMEN1
SCHEMBL22748257 0.78 MAPT (0.48) ALDH1A1MAPTGAAMEN1KMT2A
SCHEMBL22760576 0.76 MAT2A (0.41) ALDH1A1MAPTGAAHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed