SCHEMBL22806325

SCHEMBL22806325

N#CC(NC(=O)O)c1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
LMNA P02545 4/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
ALPG P10696 2/20 0.49
HTT P42858 3/20 0.47
HPGD P15428 2/20 0.47
USP2 O75604 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7598651 0.83 TSHR (0.47) ALDH1A1LMNASMN1; SMN2HTTHPGD
SCHEMBL7872426 0.81 MME (0.48) ALDH1A1LMNASMN1; SMN2ALPGHTT
SCHEMBL16563572 0.78 EPHX2 (0.44) ALDH1A1SMN1; SMN2HPGDTDP1EPHX2
SCHEMBL20490917 0.77 CES2 (0.43) ALDH1A1SMN1; SMN2HTTNPC1
SCHEMBL29582757 0.77 CTSS (0.53) ALDH1A1LMNASMN1; SMN2ALPGTDP1
SCHEMBL16563845 0.73 PDE2A (0.47) EPHX2PDE2A
SCHEMBL23000164 0.72 HTT (0.62) ALDH1A1LMNAHTTPDE2AKDM4E
SCHEMBL4451432 0.72 HTT (0.62) ALDH1A1LMNAHTTPDE2AKDM4E
SCHEMBL6174378 0.72 HTT (0.62) ALDH1A1LMNAHTTPDE2AKDM4E
SCHEMBL10978426 0.72 LMNA (0.53) ALDH1A1LMNASMN1; SMN2ALPGHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3986568-A1 BICYCLIC HETEROCYCLIC COMPOUNDS AS INHIBITORS OFBCDIN3D ACTIVITY Storm Therapeutics Ltd (GB) 2022-04-27 EP disclosed
WO-2020254831-A1 BICYCLIC HETEROCYCLIC COMPOUNDS AS INHIBITORS OFBCDIN3D ACTIVITY STORM THERAPEUTICS LTD (GB) 2020-12-24 WO disclosed