SCHEMBL22823720

SCHEMBL22823720

CCN1CNS(=O)(=O)c2cc(F)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 15/20 1.00
GRIA1 P42261 5/20 0.58
GRIA3 P42263 5/20 0.58
GRIA4 P48058 5/20 0.58
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PARK7 Q99497 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32682813 1.00 GRIA2 (1.00) GRIA2GRIA1GRIA3GRIA4CA1
SCHEMBL5359084 0.84 GRIA2 (0.73) GRIA2GRIA1GRIA3GRIA4CA1
SCHEMBL6505317 0.84 GRIA2 (0.72) GRIA2GRIA1GRIA3GRIA4CA1
SCHEMBL5184614 0.82 GRIA2 (0.70) GRIA2GRIA1GRIA3GRIA4
SCHEMBL6494353 0.82 GRIA2 (0.70) GRIA2GRIA1GRIA3GRIA4CA1
SCHEMBL6504948 0.82 GRIA2 (0.70) GRIA2GRIA1GRIA3GRIA4CA1
SCHEMBL2778320 0.82 GRIA2 (0.69) GRIA2GRIA1GRIA3GRIA4CA1
SCHEMBL28423069 0.80 GRIA2 (0.67) GRIA2GRIA1GRIA3GRIA4CA1
SCHEMBL6413657 0.80 GRIA2 (0.67) GRIA2
SCHEMBL5418711 0.78 GRIA2 (0.64) GRIA2CA1CA2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200397751-A1 Modulation of AMPA/kainate Receptors for the Treatment of Hypoglycemia VANDERKLISH PETER (US) 2020-12-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200397751-A1 Modulation of AMPA/kainate Receptors for the Treatment of Hypoglycemia GPR119, GRIK1, GRIK3 GRIA2 60/4885GRIA1 46/4885GRIA3 33/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.