SCHEMBL22858331

SCHEMBL22858331

Cn1nc(NC(=O)OC(C)(C)C)c(Br)c1CC1CC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.39
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
BCL2 P10415 5/20 0.35
BECN1 Q14457 4/20 0.35
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
DRD2 P14416 3/20 0.34
MAPK14 Q16539 1/20 0.34
BACE1 P56817 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OGFRL1 Q5TC84 1/20 0.32
FPR3 P25089 1/20 0.32
FPR2 P25090 1/20 0.32
GFER P55789 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22858337 0.78 USP30 (0.33) AAK1DRD2MAPK14
SCHEMBL16629272 0.74 MAPK14 (0.36) AAK1BCL2BECN1CTSSCTSK
SCHEMBL22858338 0.73 STK17B (0.37) AAK1
SCHEMBL22858298 0.72 MAPK14 (0.41) AAK1ALDH1A1CTSSCTSKDRD2
SCHEMBL18138239 0.67 DRD2 (0.39) AAK1KMT2AALDH1A1BCL2BECN1
SCHEMBL3304675 0.67 AAK1 (0.39) AAK1MAPK14BACE1
SCHEMBL30661581 0.67 AAK1 (0.39) AAK1MAPK14BACE1
SCHEMBL31482852 0.66 CYSLTR2 (0.45) AAK1DRD2MAPK14BACE1
SCHEMBL30896793 0.66 CYSLTR2 (0.45) AAK1DRD2MAPK14BACE1
SCHEMBL21597824 0.66 MAPK14 (0.43) DRD2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021000957-A1 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 北京国鸿生物医药科技有限公司 2021-01-07 WO disclosed