SCHEMBL16629272

SCHEMBL16629272

Cn1nc(NC(=O)OC(C)(C)C)c(Br)c1C#N

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.36
EGLN2 Q96KS0 3/20 0.34
CTSK P43235 4/20 0.33
CTSS P25774 2/20 0.33
TTK P33981 1/20 0.33
AAK1 Q2M2I8 2/20 0.33
LCK P06239 1/20 0.33
NPC1 O15118 1/20 0.32
RECQL P46063 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CTSB P07858 1/20 0.31
BCL2 P10415 1/20 0.31
BECN1 Q14457 1/20 0.31
BACE1 P56817 1/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28612240 0.86 ALDH1A1 (0.38) MAPK14RAB9ASMN1; SMN2LMNA
SCHEMBL16629232 0.75 ALDH1A1 (0.46) NPC1RAB9ASMN1; SMN2KDM4ELMNA
SCHEMBL22858331 0.74 AAK1 (0.39) MAPK14CTSKCTSSAAK1BCL2
SCHEMBL30079060 0.73 EGLN2 (0.36) MAPK14EGLN2CTSKTTKCA1
SCHEMBL16629294 0.72 CTSD (0.30) CTSSCTSB
SCHEMBL29766611 0.72
SCHEMBL16629292 0.71
SCHEMBL3304675 0.70 AAK1 (0.39) MAPK14AAK1LCKNPC1RECQL
SCHEMBL15274043 0.70 SSTR4 (0.32)
SCHEMBL30661581 0.70 AAK1 (0.39) MAPK14AAK1LCKNPC1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050989-A2 MACROCYCLIC COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES CS THERAPEUTICS INC. (US) 2015-04-09 WO disclosed