SCHEMBL22868083

SCHEMBL22868083

N=C(N)COc1ccc(C(F)(F)F)cc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 2/20 0.59
ALDH1A1 P00352 1/20 0.58
MAOB P27338 7/20 0.57
AOC3 Q16853 1/20 0.57
IDO1 P14902 2/20 0.47
KIF11 P52732 1/20 0.46
GRM4 Q14833 1/20 0.46
SIGMAR1 Q99720 1/20 0.45
PPARD Q03181 1/20 0.44
PPARA Q07869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6507086 0.81 ALDH1A1 (0.68) ALDH1A1MAOBAOC3KIF11GRM4
SCHEMBL3368887 0.79 WDR5 (0.66) WDR5MAOBIDO1
SCHEMBL20019078 0.78 MAOB (0.51) WDR5MAOBPPARA
SCHEMBL11537941 0.78 ALDH1A1 (0.63) ALDH1A1MAOBAOC3KIF11GRM4
SCHEMBL13629002 0.76 ALDH1A1 (0.49) WDR5ALDH1A1MAOBAOC3GRM4
SCHEMBL2111994 0.76 PPARD (0.68) ALDH1A1MAOBAOC3GRM4PPARD
Hydrochloric Acid SCHEMBL4433395 0.75 ALDH1A1 (0.48) ALDH1A1MAOBAOC3GRM4PPARD
SCHEMBL21360612 0.75 WDR5 (0.66) WDR5
SCHEMBL9194768 0.75 WDR5 (1.00) WDR5ALDH1A1
SCHEMBL4100035 0.75 WDR5 (0.66) WDR5MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021003295-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2021-01-07 WO disclosed