SCHEMBL22868093

SCHEMBL22868093

COc1nc(C(F)(F)F)c(OC2CCOCC2)cc1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.44
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
PDE4D Q08499 6/20 0.41
PDE4B Q07343 5/20 0.40
PDE4A P27815 4/20 0.40
PDE4C Q08493 4/20 0.40
PIK3CA P42336 4/20 0.39
TBK1 Q9UHD2 2/20 0.39
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
KAT2B Q92831 1/20 0.39
BAZ2B Q9UIF8 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.37
IKBKE Q14164 1/20 0.36
LRRK2 Q5S007 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22868088 0.85 SYK (0.41) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL22867965 0.72 ROCK2 (0.43) ROCK2ROCK1HSD17B1HSD17B2IRAK4
SCHEMBL22868089 0.71 HSD17B1 (0.58) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL10237458 0.69 TYK2 (0.41) KAT2BBAZ2BIRAK4LRRK2
SCHEMBL12970631 0.68 PARP15 (0.54) PDE4DPDE4BPDE4APDE4CTBK1
SCHEMBL24735664 0.66 PDE4D (0.54) PDE4DPDE4BPDE4APDE4C
SCHEMBL30278221 0.66 PDE4D (0.54) PDE4DPDE4BPDE4APDE4C
SCHEMBL1377003 0.66 KAT2B (0.69) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL28945888 0.65 PDE4D (0.53) PDE4DPDE4BPDE4APDE4C
SCHEMBL18669536 0.64 ROCK2 (0.55) ROCK2ROCK1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021003295-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2021-01-07 WO disclosed