SCHEMBL22869151

SCHEMBL22869151

CC(C)(C)OC(=O)NC(C(=O)O)c1csc(NS(=O)(=O)C2CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTPRB P23467 5/20 0.42
CTPS1 P17812 15/20 0.42
CTPS2 Q9NRF8 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22491644 0.88 PTPRB (0.44) PTPRBCTPS1CTPS2
SCHEMBL24088711 0.82 PTPRB (0.46) PTPRBCTPS1CTPS2
SCHEMBL22017475 0.81 PI4KB (0.42) PTPRB
SCHEMBL23452689 0.81 PTPRB (0.39) PTPRB
SCHEMBL11204633 0.81 PI4KB (0.42) PTPRB
SCHEMBL21044331 0.79 CTPS1 (0.47) CTPS1CTPS2
SCHEMBL8868383 0.78 CTSK (0.39) PTPRB
SCHEMBL21044563 0.78 CTPS1 (0.43) CTPS1CTPS2
SCHEMBL5967488 0.77 PTPRB (0.52) PTPRB
SCHEMBL24088721 0.77 CTPS1 (0.42) PTPRBCTPS1CTPS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3717459-B1 COMPOUNDS STEP PHARMA S A S (FR) 2026-01-21 EP disclosed
EP-4232425-A1 CTPS1 INHIBITORS AND USES THEREOF Nimbus Clotho, Inc. (US) 2023-08-30 EP disclosed
CN-116601131-A CTPS1 inhibitor and application thereof 林伯士克洛索有限公司 2023-08-15 CN disclosed
US-11655246-B2 Aminothiazole compounds as inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2023-05-23 US disclosed
US-11655246-B2 Aminothiazole compounds as inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2023-05-23 US disclosed
US-20230077316-A1 CTPS1 INHIBITORS AND USES THEREOF NIMBUS DISCOVERY, INC. 2023-03-09 US disclosed
WO-2022087634-A1 CTPS1 INHIBITORS AND USES THEREOF NIMBUS CLOTHO, INC. (US) 2022-04-28 WO disclosed
WO-2022087634-A1 CTPS1 INHIBITORS AND USES THEREOF NIMBUS CLOTHO, INC. (US) 2022-04-28 WO disclosed
US-20210002269-A1 COMPOUNDS STEP PHARMA S.A.S. (FR) 2021-01-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11655246-B2 Aminothiazole compounds as inhibitors of CTPS1 CTPS1, CTPS2, TBXAS1 PTPRB 3195/4885CTPS1 1/4885CTPS2 2/4885
US-20230077316-A1 CTPS1 INHIBITORS AND USES THEREOF CTPS1, CTPS2, ECHS1 PTPRB 2590/4885CTPS1 1/4885CTPS2 2/4885
US-20210002269-A1 COMPOUNDS UGT1A1, CYP1A1, CYP19A1 PTPRB 4627/4885CTPS1 2385/4885CTPS2 2441/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.