9-Methylguanine

9-Methylguanine

SCHEMBL22884

Cn1cnc2c(=O)[nH]c(N)nc21

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
XDH P47989 8/20 0.58
TK1 P04183 2/20 0.57
PNP P00491 4/20 0.54
USP2 O75604 1/20 0.52
TSHR P16473 1/20 0.52
EDNRA P25101 1/20 0.52
HTR2A P28223 1/20 0.52
RECQL P46063 1/20 0.52
BLM P54132 1/20 0.52
HBB P68871 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HPRT1 P00492 4/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
9-Methylguanine SCHEMBL27339404 0.98 XDH (0.57) XDHTK1PNPUSP2TSHR
9-Methylguanine SCHEMBL27638388 0.90 XDH (0.52) XDHTK1PNPUSP2TSHR
9-Methylguanine SCHEMBL28106048 0.83 XDH (0.47) XDHTK1PNPUSP2TSHR
SCHEMBL986800 0.82 XDH (0.60) XDHTK1PNPUSP2TSHR
SCHEMBL29286376 0.81 TK1 (0.76) TK1PNPUSP2TSHREDNRA
SCHEMBL41787 0.81 XDH (0.59) XDHTK1PNPUSP2TSHR
SCHEMBL27667185 0.81 XDH (0.63) XDHTK1PNPUSP2TSHR
SCHEMBL9910656 0.81 XDH (0.42) XDHTK1PNPHPRT1KMT2A
SCHEMBL15005119 0.81 XDH (0.59) XDHTK1PNPUSP2TSHR
SCHEMBL24374442 0.80 XDH (0.47) XDHTK1PNPHPRT1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6169 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026099790-A1 DEVICE USING ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2026-05-15 WO claimed
US-20260131157-A1 METHODS OF USING ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2026-05-14 US claimed
US-20260115161-A1 2-HYDROXY-OCTADECENE-9-CIS-OATE FOR USE IN THE TREATMENT OF ONCOLOGICAL PATHOLOGIES AND NEUROPATHIC PAIN LAMINAR PHARMACEUTICALS S A (ES) 2026-04-30 US claimed
US-12569572-B2 Messenger RNA therapy for the treatment of Friedreich's ataxia TRANSLATE BIO, INC. (US) 2026-03-10 US claimed
EP-4663187-A1 2-HYDROXY-OCTADECENE-9-CIS-OATE FOR USE IN THE TREATMENT OF ONCOLOGICAL PATHOLOGIES AND NEUROPATHIC PAIN Laminar Pharmaceuticals, S.A. (ES) 2025-12-17 EP claimed
EP-4452256-B1 METHODS OF TREATING BRAIN TUMOURS AND NEUROBLASTOMAS ASTRAZENECA AB (SE) 2025-12-10 EP claimed
US-12473663-B2 Compositions and methods for immune repertoiresequencing Life Technologies Corporation (US) 2025-11-18 US claimed
US-20250312347-A1 THERAPEUTIC BENEFIT OF SUBOPTIMALLY ADMINISTERED CHEMICAL COMPOUNDS BROWN DENNIS M (US) 2025-10-09 US claimed
EP-4267763-B1 COMPOSITIONS AND METHODS FOR HIGHLY SENSITIVE DETECTION OF TARGET SEQUENCES IN MULTIPLEX REACTIONS LIFE TECHNOLOGIES CORP (US) 2025-07-23 EP claimed
US-12350318-B2 Combination therapy to treat brain cancer INOVIO PHARMACEUTICALS, INC. (US) 2025-07-08 US claimed
WO-2000058329-A1 CLEAVAGE OF NUCLEIC ACID FROM SOLID SUPPORTS GOLDSBOROUGH, ANDREW (FR) 2000-10-05 WO claimed
WO-1999025386-A1 delta-O6-METHYLGUANINE-DNA METHYLTRANSFERASE GENE TRANSFER FOR O6-BENZYLGUANINE AND (N,N'-BIS(2-CHLOROETHYL)-N-NITROSOUREA) RESISTANCE CASE WESTERN RESERVE UNIVERSITY (US) 1999-05-27 WO claimed
WO-1998042723-A9 METHODS AND COMPOSITIONS FOR THE DIAGNOSIS AND TREATMENT OF NEUROPSYCHIATRIC DISORDERS 1999-03-04 WO claimed
EP-0540693-B1 THE REDUCTION OF NON-SPECIFIC AMPLIFICATION DURING $i(IN VITRO) NUCLEIC ACID AMPLIFICATION USING MODIFIED NUCLEIC ACID BASES HOFFMANN LA ROCHE (CH) 1999-01-20 EP claimed
US-5703224-A Antiviral c-nucleoside derivatives NIPPON SHINYAKU CO. LTD. (JP) 1997-12-30 US claimed
EP-0733630-A1 NUCLEOSIDE DERIVATIVE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1996-09-25 EP claimed
EP-0625985-A1 METHOD AND RING-OPENED PURINE COMPOUNDS FOR LABELING POLYNUCLEOTIDES. UNIV MIAMI (US) 1994-11-30 EP claimed
WO-1993011146-A1 METHOD AND RING-OPENED PURINE COMPOUNDS FOR LABELING POLYNUCLEOTIDES UNIVERSITY OF MIAMI (US) 1993-06-10 WO claimed
EP-0540693-A1 THE REDUCTION OF NON-SPECIFIC AMPLIFICATION DURING $i(IN VITRO) NUCLEIC ACID AMPLIFICATION USING MODIFIED NUCLEIC ACID BASES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1993-05-12 EP claimed
WO-1992001814-A2 THE REDUCTION OF NON-SPECIFIC AMPLIFICATION DURING IN VITRO NUCLEIC ACID AMPLIFICATION USING MODIFIED NUCLEIC ACID BASES F. HOFFMANN-LA-ROCHE AG (CH) 1992-02-06 WO claimed