SCHEMBL22890853

SCHEMBL22890853

Nc1ccc2c(c1)c(C(F)F)nn2C1CCCCO1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RET P07949 7/20 0.37
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
CYP4F2 P78329 2/20 0.35
CYP4A11 Q02928 2/20 0.35
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ATR Q13535 6/20 0.32
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29643967 1.00 RET (0.37) RETRXRARXRBRXRGCYP4F2
SCHEMBL21198696 0.84 CYP4F2 (0.39) RETRXRARXRBRXRGCYP4F2
SCHEMBL21217456 0.83 RET (0.37) RETRXRARXRBRXRGCYP4F2
SCHEMBL31422772 0.82 CYP1A2 (0.38) RXRARXRBRXRGALDH1A1LMNA
SCHEMBL24610343 0.81 GAA (0.47) RETRXRARXRBRXRGCYP4F2
SCHEMBL21198529 0.81 GAA (0.47) RETRXRARXRBRXRGCYP4F2
SCHEMBL29388171 0.81 ALDH1A1 (0.39) RETRXRARXRBRXRGCYP4F2
SCHEMBL14863556 0.81 ALDH1A1 (0.39) RETRXRARXRBRXRGCYP4F2
SCHEMBL22890826 0.81 RXRA (0.37) RETRXRARXRBRXRGCYP4F2
SCHEMBL22889886 0.81 RET (0.40) RETRXRARXRBRXRGCYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021007477-A1 INDAZOLES AND AZAINDAZOLES AS LRRK2 INHIBITORS E-SCAPE BIO, INC. (US) 2021-01-14 WO disclosed