SCHEMBL22908712

SCHEMBL22908712

O=C1CC(c2ccc([N+](=O)[O-])cc2)=NN1c1ccc(Cl)cc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.60
MAPT P10636 7/20 0.60
MEN1 O00255 6/20 0.60
LMNA P02545 1/20 0.60
L3MBTL1 Q9Y468 2/20 0.56
GAA P10253 2/20 0.56
NPSR1 Q6W5P4 1/20 0.56
CD274 Q9NZQ7 4/20 0.46
PDCD1 Q15116 3/20 0.46
MAPK1 P28482 1/20 0.45
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HPGD P15428 1/20 0.44
GABRA2 P47869 1/20 0.43
GABRB2 P47870 1/20 0.43
POLB P06746 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
PGR P06401 1/20 0.42
KDM4E B2RXH2 2/20 0.41
HTT P42858 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22908674 0.87 KMT2A (0.70) KMT2AMAPTMEN1LMNAGAA
SCHEMBL10435326 0.82 MAPT (0.75) KMT2AMAPTMEN1LMNAL3MBTL1
SCHEMBL22908646 0.80 KMT2A (0.61) KMT2AMAPTMEN1LMNAGAA
SCHEMBL22908683 0.75 KMT2A (0.58) KMT2AMAPTMEN1LMNAGAA
SCHEMBL10435508 0.75 MEN1 (0.67) KMT2AMAPTMEN1LMNAL3MBTL1
SCHEMBL22909309 0.75 KMT2A (0.55) KMT2AMAPTMEN1LMNAGAA
SCHEMBL10435116 0.75 MAPT (0.90) KMT2AMAPTMEN1LMNAL3MBTL1
SCHEMBL11182553 0.74 PDCD1 (0.56) KMT2AMAPTMEN1LMNAL3MBTL1
SCHEMBL22909301 0.74 KMT2A (0.62) KMT2AMAPTMEN1LMNAGAA
SCHEMBL22909489 0.72 CD274 (0.57) KMT2AMAPTMEN1LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3766544-A1 NOVEL PYRAZOLONE DERIVATIVES AS PD-1/PD-L1 INTERACTION INHIBITORS Centre Hospitalier Regional Universitaire de Lille (FR) 2021-01-20 EP disclosed