SCHEMBL22909451

SCHEMBL22909451

CN(C)S(=O)(=O)c1c(F)c(F)c(F)c(F)c1OCc1ccc(C#N)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.40
MAOB P27338 9/20 0.39
ACHE P22303 3/20 0.38
MAOA P21397 2/20 0.38
SMPD1 P17405 1/20 0.37
NSD2 O96028 1/20 0.36
CYP19A1 P11511 1/20 0.36
AR P10275 1/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22909373 0.83 AR (0.45) NPC1RAB9ACYP19A1AR
SCHEMBL22909262 0.81 HDAC6 (0.39) NPC1RAB9AMAOBALOX5APFEN1
SCHEMBL29729050 0.81 HDAC6 (0.39) NPC1RAB9AMAOBALOX5APFEN1
SCHEMBL29671227 0.79 CYP19A1 (0.50) MAOBCYP19A1
SCHEMBL22909344 0.79 PARP10 (0.48) TSHRMAOBALOX5APFEN1
SCHEMBL29671275 0.75 CA2 (0.48) TSHRNPC1NSD2CYP19A1
SCHEMBL29729048 0.72 CA1 (0.31)
SCHEMBL22909160 0.72 MAPT (0.36) TSHR
SCHEMBL22909484 0.71 CA1 (0.40) TSHR
SCHEMBL22909370 0.71 SMN1; SMN2 (0.43) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12559454-B2 Benzenesulfonamide derivatives and uses thereof 2692372 ONTARIO, INC. (CA) 2026-02-24 US disclosed
US-20220281812-A1 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 ONTARIO INC (CA) 2022-09-08 US disclosed
EP-4017843-A1 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 Ontario, Inc. (CA) 2022-06-29 EP disclosed
CN-114502533-A Benzenesulfonamide derivatives and use thereof 2692372安大略公司 2022-05-13 CN disclosed
WO-2021009568-A1 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 ONTARIO, INC. (CA) 2021-01-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12559454-B2 Benzenesulfonamide derivatives and uses thereof NR2E1, NR2C2, NR3C1 TSHR 39/4885NPC1 272/4885RAB9A 2966/4885
US-20220281812-A1 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF BCR, ARSA, VHL TSHR 2336/4885NPC1 1221/4885RAB9A 2441/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.