SCHEMBL22915969

SCHEMBL22915969

Cc1cccc(C(=O)N2CCc3[nH]cnc3C2)c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.51
CDK4 P11802 4/20 0.50
CCND1 P24385 4/20 0.50
GRM5 P41594 3/20 0.48
GABRD O14764 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB1 P18505 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GABRA2 P47869 1/20 0.46
GABRB2 P47870 1/20 0.46
GABRA4 P48169 1/20 0.46
NAMPT P43490 1/20 0.46
HTR2C P28335 1/20 0.46
KDM4E B2RXH2 2/20 0.45
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CYP3A4 P08684 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20214414 0.86 SMN1; SMN2 (0.57) HPGDCDK4CCND1GRM5GABRA1
SCHEMBL22915971 0.86 SLC6A7 (0.52) HPGDCDK4CCND1NAMPTHTR2C
SCHEMBL20214653 0.86 GRM5 (0.50) HPGDGRM5NAMPTKDM4EL3MBTL1
SCHEMBL22916015 0.85 POLB (0.57) HPGDNAMPTHTR2CKDM4EHTT
SCHEMBL22916012 0.85 ALDH1A1 (0.53) HPGDCDK4CCND1GRM5L3MBTL1
SCHEMBL22915970 0.85 POLB (0.55) HPGDCDK4CCND1GRM5GABRD
SCHEMBL22915890 0.85 KDM4E (0.47) HPGDGRM5NAMPTHTR2CKDM4E
SCHEMBL22915942 0.82 GRM5 (0.50) HPGDCDK4CCND1GRM5NAMPT
SCHEMBL20214648 0.82 KMT2A (0.47) HPGDCDK4CCND1GRM5NAMPT
SCHEMBL22915886 0.81 NAMPT (0.51) HPGDGRM5NAMPTHTR2CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3548613-B1 BACTERIAL GLUTAMINYL CYCLASE INHIBITORS AND USE THEREOF IN THE TREATMENT OF PERIODONTITIS FRAUNHOFER GES FORSCHUNG (DE) 2021-01-27 EP disclosed