SCHEMBL22916246

SCHEMBL22916246

CCN[C@@H]1c2ccccc2C[C@H]1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.47
SLC6A3 Q01959 1/20 0.47
MAOB P27338 3/20 0.45
MAOA P21397 2/20 0.45
MMP1 P03956 4/20 0.45
MMP2 P08253 4/20 0.45
MMP9 P14780 4/20 0.45
MMP8 P22894 4/20 0.45
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
OPRM1 P35372 1/20 0.42
OPRK1 P41145 1/20 0.42
NAMPT P43490 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8437280 1.00 SLC6A4 (0.47) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL21916845 1.00 SLC6A4 (0.47) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL12472928 1.00 SLC6A4 (0.47) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL13256435 1.00 SLC6A4 (0.47) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL23330350 0.87 SIGMAR1 (0.50) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL23420183 0.83 MMP9 (0.52) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL22062447 0.82 SLC6A4 (0.44) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL13283348 0.82 MAOB (0.68) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL8279734 0.80 MEN1 (0.46) SLC6A4SLC6A3MAOBMAOAMMP1
SCHEMBL1239662 0.80 MEN1 (0.46) SLC6A4SLC6A3MAOBMAOAMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11992494-B2 Cyclopentathiophene carboxamide derivatives as platelet activating factor receptor antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-05-28 US disclosed
US-20230190763-A1 Cyclopentathiophene Carboxamide Derivatives as Platelet Activating Factor Receptor Antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-22 US disclosed
US-20210024462-A1 SULFAMOYL-ARYLAMIDES AND THE USE THEREOF AS MEDICAMENTS FOR THE TREATMENT OF HEPATITIS B JANSSEN SCIENCES IRELAND UNLIMITED CO (IE) 2021-01-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11992494-B2 Cyclopentathiophene carboxamide derivatives as platelet activating factor receptor antagonists PTAFR, PDGFRA, PDGFRB SLC6A4 2427/4885SLC6A3 3321/4885MAOB 3041/4885
US-20230190763-A1 Cyclopentathiophene Carboxamide Derivatives as Platelet Activating Factor Receptor Antagonists PTAFR, PDGFRA, PDGFRB SLC6A4 2427/4885SLC6A3 3321/4885MAOB 3041/4885
US-20210024462-A1 SULFAMOYL-ARYLAMIDES AND THE USE THEREOF AS MEDICAMENTS FOR THE TREATMENT OF HEPATITIS B SULT2A1, HCCS, SULT1A1 SLC6A4 3343/4885SLC6A3 4239/4885MAOB 1293/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.