SCHEMBL22916892

SCHEMBL22916892

CC(C)NC(=O)CCNC(=O)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
FAAH O00519 1/20 0.47
MAPK1 P28482 1/20 0.47
EPHX2 P34913 1/20 0.41
EPHX1 P07099 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ECE1 P42892 3/20 0.39
ALDH1A1 P00352 3/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 2/20 0.35
USP2 O75604 1/20 0.35
KDM4E B2RXH2 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TERT O14746 1/20 0.35
CHRM5 P08912 1/20 0.34
CHRM3 P20309 1/20 0.34
DPP4 P27487 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25532290 0.88 KMT2A (0.53) KMT2AMEN1FAAHMAPK1EPHX2
SCHEMBL861045 0.85 KMT2A (0.46) KMT2AMEN1FAAHMAPK1EPHX2
SCHEMBL25532300 0.82 KMT2A (0.51) KMT2AMEN1FAAHMAPK1EPHX2
SCHEMBL23011663 0.81 MAPK1 (0.48) KMT2AMEN1FAAHMAPK1EPHX2
SCHEMBL22917270 0.81 EPHX1 (0.55) KMT2AMEN1MAPK1EPHX2EPHX1
SCHEMBL12734811 0.81 LMNA (0.41) KMT2AMEN1MAPK1CYP2D6CYP2C9
SCHEMBL19901903 0.81 KMT2A (0.54) KMT2AMEN1FAAHMAPK1EPHX2
SCHEMBL861319 0.81 KMT2A (0.54) KMT2AMEN1FAAHMAPK1EPHX2
SCHEMBL21128132 0.79 ALDH1A1 (0.41) KMT2AMEN1MAPK1CYP2D6CYP2C9
SCHEMBL13853860 0.79 KMT2A (0.47) KMT2AMEN1FAAHMAPK1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230159554-A1 COMPOUND WITH ANTICANCER ACTIVITY KYOWA KIRIN CO., LTD. (JP) 2023-05-25 US disclosed
US-20230159554-A1 COMPOUND WITH ANTICANCER ACTIVITY KYOWA KIRIN CO., LTD. (JP) 2023-05-25 US disclosed
US-20230150974-A1 COMPOUNDS AND USES THEREOF FOGHORN THERAPEUTICS INC. 2023-05-18 US disclosed
EP-3778573-A1 COMPOUND WITH ANTICANCER ACTIVITY Kyowa Kirin Co., Ltd. (JP) 2021-02-17 EP disclosed
US-20210024540-A1 COMPOUND WITH ANTICANCER ACTIVITY KYOWA KIRIN CO., LTD. (JP) 2021-01-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210024540-A1 COMPOUND WITH ANTICANCER ACTIVITY TP53, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, RCC2 KMT2A 2349/4885MEN1 41/4885FAAH 4699/4885
US-20230150974-A1 COMPOUNDS AND USES THEREOF VHL, CLN6, TFEB KMT2A 792/4885MEN1 1366/4885FAAH 3729/4885
US-20230159554-A1 COMPOUND WITH ANTICANCER ACTIVITY TP53, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, RCC2 KMT2A 2349/4885MEN1 41/4885FAAH 4699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.