SCHEMBL22923901

SCHEMBL22923901

Cc1ccnc2[nH]cc(-c3ccccc3)c12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 10/20 0.54
ROCK1 Q13464 8/20 0.51
PRKACA P17612 6/20 0.51
CDK5 Q00535 6/20 0.51
DYRK1A Q13627 6/20 0.51
PRKD3 O94806 5/20 0.51
MAP4K4 O95819 5/20 0.51
CLK2 P49760 5/20 0.51
MAP4K2 Q12851 5/20 0.51
GSK3A P49840 5/20 0.51
GSK3B P49841 5/20 0.51
NTRK3 Q16288 4/20 0.51
PAK4 O96013 4/20 0.51
CDK8 P49336 4/20 0.51
CLK4 Q9HAZ1 4/20 0.51
NTRK2 Q16620 4/20 0.51
NTRK1 P04629 4/20 0.51
MAP2K1 Q02750 3/20 0.51
CAMK2A Q9UQM7 3/20 0.51
TAOK1 Q7L7X3 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22096096 0.80 LRRK2 (0.50) LRRK2ROCK1PRKACACDK5DYRK1A
SCHEMBL29952060 0.80 LRRK2 (0.50) LRRK2ROCK1PRKACACDK5DYRK1A
SCHEMBL29952435 0.78 LRRK2 (0.51) LRRK2ROCK1PRKACACDK5DYRK1A
SCHEMBL855137 0.76 HTR2A (0.48) LRRK2ROCK1CDK5JAK3CDK9
SCHEMBL13045933 0.75 NPC1 (0.48) LRRK2ROCK1PRKACACDK5DYRK1A
SCHEMBL3740263 0.74 CAMKK2 (0.69) LRRK2ROCK1PRKACACDK5DYRK1A
SCHEMBL14462648 0.73 LRRK2 (0.61) LRRK2ROCK1PRKACACDK5DYRK1A
SCHEMBL4790325 0.73 LRRK2 (0.61) LRRK2ROCK1PRKACACDK5DYRK1A
SCHEMBL4790877 0.73 LRRK2 (0.61) LRRK2ROCK1PRKACACDK5DYRK1A
SCHEMBL29953748 0.73 LRRK2 (0.57) LRRK2ROCK1PRKACACDK5DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021012717-A1 ANTITUMOR COMPOUND USED AS AXL INHIBITOR AND USE THEREOF 南京华威医药科技集团有限公司 2021-01-28 WO disclosed