SCHEMBL22927677

SCHEMBL22927677

CCOc1c(C(=O)O)nc(N(C)Cc2ccc(Cl)cc2)n(C)c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 4/20 0.37
KLKB1 P03952 1/20 0.37
ALDH1A1 P00352 5/20 0.37
HTT P42858 2/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 2/20 0.36
MAPK1 P28482 3/20 0.35
TSHR P16473 2/20 0.35
HDAC6 Q9UBN7 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
HSD17B10 Q99714 2/20 0.35
ALOX15 P16050 1/20 0.35
POLB P06746 1/20 0.35
KDM4E B2RXH2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ABCB1 P08183 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22927731 0.90 MAPK1 (0.43) ALDH1A1HTTNPSR1MAPK1TSHR
SCHEMBL22927759 0.88 KMT2A (0.43) ALDH1A1HTTHDAC6MAOAMAOB
SCHEMBL22927760 0.88 KCNH2 (0.39) HTTNPSR1KDM4ESMN1; SMN2MEN1
SCHEMBL22927803 0.88 HDAC6 (0.38) ALDH1A1HTTRAB9ANPSR1MAPK1
SCHEMBL22927765 0.87 MEN1 (0.35) ALDH1A1RAB9AMAOBSMN1; SMN2MEN1
SCHEMBL22927766 0.86 COPS5 (0.36) ALDH1A1HTTNPSR1TSHRALOX15
SCHEMBL29434810 0.81 LMNA (0.43) ALDH1A1HTTNPSR1MAPK1TSHR
SCHEMBL22927753 0.80 HDAC6 (0.38) F10ALDH1A1RAB9ANPSR1MAPK1
SCHEMBL22927770 0.80 NR3C1 (0.41) ALDH1A1HTTNPSR1MAPK1TSHR
SCHEMBL22927676 0.80 MAOB (0.51) ALDH1A1RAB9ANPSR1MAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021016317-A1 MODULATORS OF TREX1 CONSTELLATION PHARMACEUTICALS, INC. (US) 2021-01-28 WO disclosed