SCHEMBL22928459

SCHEMBL22928459

COc1nccc(O)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.37
NOS3 P29474 2/20 0.36
NOS2 P35228 2/20 0.36
NOS1 P29475 1/20 0.36
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.34
HPGD P15428 2/20 0.34
APLNR P35414 1/20 0.34
MAPK1 P28482 2/20 0.33
AURKA O14965 1/20 0.33
TTK P33981 1/20 0.33
AURKB Q96GD4 1/20 0.33
INCENP Q9NQS7 1/20 0.33
TRPA1 O75762 1/20 0.33
ATM Q13315 1/20 0.33
MTNR1A P48039 1/20 0.33
TLR8 Q9NR97 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17946845 0.78 NOS3 (0.36) CYP3A4NOS3NOS2NOS1CCR1
SCHEMBL30975066 0.78 TDP1 (0.38) CYP3A4NOS3NOS2NOS1CCR1
SCHEMBL21552375 0.78 TDP1 (0.38) CYP3A4NOS3NOS2NOS1CCR1
SCHEMBL6792963 0.77 NOS3 (0.48) NOS3NOS2NOS1CCR1CCR5
SCHEMBL16618427 0.77 NOS3 (0.35) CYP3A4NOS3NOS2NOS1CCR1
SCHEMBL10201420 0.77 NOS3 (0.35) CYP3A4NOS3NOS2NOS1CCR1
SCHEMBL31289813 0.77 HPGD (0.40) CYP3A4NOS3NOS2NOS1CCR1
SCHEMBL4074890 0.76 ALDH1A1 (0.44) CYP3A4CCR1CCR5CCR8ALDH1A1
SCHEMBL18686676 0.75 ENPP2 (0.36) NOS3NOS2NOS1CCR1CCR5
SCHEMBL22972330 0.74 TRPA1 (0.37) CYP3A4NOS3NOS2NOS1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3380101-B1 EIF4-A-INHIBITING COMPOUNDS AND METHODS RELATED THERETO EFFECTOR THERAPEUTICS INC (US) 2021-01-27 EP disclosed