SCHEMBL2293261

SCHEMBL2293261

CCOC(=O)Cc1c(F)ccc2cnc(OC)nc12

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.39
MAOB P27338 3/20 0.38
KDM4E B2RXH2 4/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPK1 P28482 2/20 0.36
HSD17B10 Q99714 2/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36
DPP4 P27487 2/20 0.35
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2292326 0.78 ALDH1A1 (0.34) KDM4EL3MBTL1TDP1MEN1MAPT
SCHEMBL1723475 0.75 KCNH2 (0.42) MAOBKDM4ESMN1; SMN2ALDH1A1
SCHEMBL2285150 0.74 ALDH1A1 (0.34) KDM4EL3MBTL1TDP1MAPTKMT2A
SCHEMBL2293987 0.72 ALDH1A1 (0.34) L3MBTL1TDP1MEN1MAPTKMT2A
SCHEMBL3411112 0.72 PTGS2 (0.46) PTGS2KDM4EL3MBTL1MAPTHSD17B10
SCHEMBL1711837 0.71 PTGS2 (0.55) PTGS2
SCHEMBL7494802 0.71 NLRP3 (0.42) KDM4EL3MBTL1TDP1MEN1MAPT
SCHEMBL31618210 0.70 HPGD (0.49) KDM4EL3MBTL1TDP1MEN1MAPT
SCHEMBL23485370 0.70 SMN1; SMN2 (0.46) MAOBKDM4EL3MBTL1MAPTSMN1; SMN2
SCHEMBL1867904 0.69 NLRP3 (0.54) KDM4EL3MBTL1TDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8618092-B2 Tricyclic oxazolidinone antibiotic compounds ACTELION PHARMACEUTICALS LTD. (CH) 2013-12-31 US disclosed
US-20110195961-A1 TRICYCLIC OXAZOLIDINONE ANTIBIOTIC COMPOUNDS ACTELION PHARMACEUTICALS LTD. (CH) 2011-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110195961-A1 TRICYCLIC OXAZOLIDINONE ANTIBIOTIC COMPOUNDS HRH3, OXA1L, HRH1 PTGS2 4023/4885MAOB 2979/4885KDM4E 3061/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.