SCHEMBL22945945

SCHEMBL22945945

COC(=O)c1cccc2[nH]c(-c3ccc(CN(C)C(=O)OC(C)(C)C)cc3)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 1/20 0.42
TNKS O95271 4/20 0.39
CSF1R P07333 3/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
CTSV O60911 1/20 0.38
CTSL P07711 1/20 0.38
PARP1 P09874 2/20 0.37
GLS O94925 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
CACNA1G O43497 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1C Q13936 1/20 0.35
LTB4R2 Q9NPC1 1/20 0.35
NR4A2 P43354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22946038 0.82 HDAC11 (0.40) HDAC11CSF1RALDH1A1CDK5CDK5R1
SCHEMBL4776229 0.78 AOC3 (0.43) CSF1RALDH1A1GLSCHUKINSR
SCHEMBL22945943 0.77 ALDH1A1 (0.36) ALDH1A1MAPTPARP1GLSHDAC3
SCHEMBL4406811 0.77 TNKS (0.38) HDAC11TNKSCSF1RALDH1A1MAPT
SCHEMBL22946360 0.76 RIPK1 (0.36) CSF1RALDH1A1CACNA1GCACNA1BCACNA1C
SCHEMBL5002616 0.75 SLC6A4 (0.52) HDAC11ALDH1A1MAPTCDK5CDK5R1
SCHEMBL30964962 0.74 GLS (0.40) ALDH1A1MAPTCTSLGLSCACNA1G
SCHEMBL8266460 0.73 TNKS (0.39) TNKSCSF1RALDH1A1MAPTPARP1
SCHEMBL27636818 0.73 CTSV (0.44) HDAC11CSF1RALDH1A1CDK5CDK5R1
SCHEMBL22300790 0.72 NAMPT (0.42) HDAC11PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021018298-A1 INDOLO-SEVEN-MEMBERED ACYLOXIME COMPOUNDS AS PARP INHIBITORS 南京明德新药研发有限公司 2021-02-04 WO disclosed