SCHEMBL22959296

SCHEMBL22959296

COc1ccc(CS)nc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.48
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
MBOAT4 Q96T53 1/20 0.40
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
TUBB4A P04350 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1581469 0.81 PDE10A (0.43) CA12CA1CA2CA7CA9
SCHEMBL29723725 0.79 P2RX7 (0.45) CA12CA1CA2CA7CA9
SCHEMBL29987012 0.79 ALDH1A1 (0.44) CA12CA1CA2CA7CA9
SCHEMBL29723727 0.79 P2RX7 (0.45) CA12CA1CA2CA7CA9
SCHEMBL10002478 0.79 MAOB (0.43) IDO1CA12CA1CA2CA7
SCHEMBL5032709 0.79 CA12 (0.40) CA12CA1CA2CA7CA9
SCHEMBL30015156 0.79 CA12 (0.40) CA12CA1CA2CA7CA9
SCHEMBL21909726 0.79 CA12 (0.40) CA12CA1CA2CA7CA9
SCHEMBL19432655 0.79 MBOAT4 (0.43) CA12CA1CA2CA7CA9
SCHEMBL731990 0.79 P2RX7 (0.45) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023280073-A1 METHOD FOR PREPARING NITROGEN-CONTAINING POLYCYCLIC FUSED RING COMPOUND, AND INTERMEDIATE AND USE OF COMPOUND 北京志健金瑞生物医药科技有限公司 2023-01-12 WO disclosed
WO-2021023209-A1 NITROGEN-CONTAINING POLYCYCLIC FUSED RING COMPOUNDS, AND PHARMACEUTICAL COMPOSITION THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 北京志健金瑞生物医药科技有限公司 2021-02-11 WO disclosed