SCHEMBL22968427

SCHEMBL22968427

O=C(O)c1cnn(-c2cccc(F)c2C(=O)O)n1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 17/20 0.40
HCRTR2 O43614 16/20 0.40
PLAU P00749 1/20 0.38
ELANE P08246 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
ADAMTS7 Q9UKP4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23354698 0.87 ADAMTS7 (0.38) HCRTR1HCRTR2PLAUELANECES2
SCHEMBL23354796 0.86 ADAMTS7 (0.47) ADAMTS7
SCHEMBL29597179 0.83 HCRTR1 (0.49) HCRTR1HCRTR2CES2CES1
SCHEMBL1586205 0.83 HCRTR1 (0.49) HCRTR1HCRTR2CES2CES1
SCHEMBL15639716 0.81 KDM4E (0.38) HCRTR1HCRTR2PLAUELANECES2
Iodomethane SCHEMBL31482883 0.79 HCRTR1 (0.48) HCRTR1HCRTR2
SCHEMBL23354732 0.75 KMO (0.38) CES2CES1ADAMTS7
SCHEMBL23354661 0.75 KMO (0.41) CES2CES1
SCHEMBL23354899 0.74 ALDH1A1 (0.52)
SCHEMBL23354846 0.74 ADORA2A (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021023843-A1 IMPROVED SYNTHETIC METHODS OF MAKING (2H-1,2,3-TRIAZOL-2-YL)PHENYL COMPOUNDS AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2021-02-11 WO disclosed