SCHEMBL22972377

SCHEMBL22972377

CCc1ccnc(C(=O)N2CCC(F)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.49
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
CSF1R P07333 3/20 0.40
HRH3 Q9Y5N1 3/20 0.39
MGLL Q99685 1/20 0.39
SLC6A7 Q99884 1/20 0.38
EPHX2 P34913 1/20 0.38
MAP3K12 Q12852 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
DPP4 P27487 1/20 0.38
HPGD P15428 1/20 0.38
RBP4 P02753 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL805504 0.86 SMYD3 (0.47) SMYD3L3MBTL1CSF1RSLC6A7NPC1
SCHEMBL11918962 0.85 SMN1; SMN2 (0.49) SMYD3CSF1RNPC1RAB9AHPGD
SCHEMBL11919148 0.82 CFTR (0.45) SMYD3L3MBTL1CSF1RHPGD
SCHEMBL22972208 0.74 L3MBTL1 (0.75) L3MBTL1EPHX2HPGDRBP4
SCHEMBL2677778 0.73 SMYD3 (0.54) SMYD3L3MBTL1NPC1RAB9A
SCHEMBL22840323 0.72 NPC1 (0.50) L3MBTL1HRH3NPC1RAB9AHPGD
SCHEMBL25187614 0.72 HRH3 (0.35) SMYD3HCRTR1HCRTR2CSF1RHRH3
SCHEMBL12257113 0.72 RAB9A (0.50) NPC1RAB9AHPGD
SCHEMBL221963 0.71 ALDH1A1 (0.55) SMYD3L3MBTL1
SCHEMBL6173009 0.71 SMYD3 (0.51) SMYD3L3MBTL1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021023888-A1 ISOQUINOLINE DERIVATIVES AS PROTEIN KINASE INHIBITORS B.C.I. PHARMA (BE) 2021-02-11 WO disclosed