SCHEMBL2299690

SCHEMBL2299690

O=C(O)c1c(Cl)nc2c(c1O)C(=O)CC1(CCC1)C2

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.34
PIK3CD O00329 2/20 0.32
PIK3CA P42336 2/20 0.32
PIK3CB P42338 2/20 0.32
PIK3CG P48736 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2303992 0.86 PIK3CD (0.30) CYP11B2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL661613 0.71 CYP1A2 (0.43)
SCHEMBL16258372 0.69 LMNA (0.37)
SCHEMBL663100 0.69 CYP1A2 (0.43)
SCHEMBL664932 0.66 PIK3CD (0.36) CYP11B2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16931070 0.60 NTRK3 (0.39)
SCHEMBL6492773 0.57 POLB (0.48)
SCHEMBL29841493 0.55 ALDH1A1 (0.43)
SCHEMBL28867137 0.55 ALDH1A1 (0.43)
SCHEMBL1989330 0.54 ALDH1A1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536733-A1 TRICYCLIC PYRIDINE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PREPARATION Boehringer Ingelheim International GmbH (DE) 2012-12-26 EP disclosed
WO-2011101424-A1 TRICYCLIC PYRIDINE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PREPARATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-25 WO disclosed