SCHEMBL23006099

SCHEMBL23006099

CC(C)[C@@H](C)c1cccc(C2CN(C)C2)n1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
KCNH2 Q12809 1/20 0.33
CHRNA7 P36544 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23106870 0.87 CHRNA7 (0.42) HTR1ADRD2DRD4KCNH2CHRNA7
SCHEMBL23006101 0.76 TLR9 (0.38)
SCHEMBL23114604 0.73 TGFBR1 (0.33) KCNH2
SCHEMBL23103376 0.73 DRD2 (0.43) DRD2KCNH2
SCHEMBL23103374 0.73 DRD2 (0.43) DRD2KCNH2
SCHEMBL23103365 0.73 DRD2 (0.43) DRD2KCNH2
SCHEMBL29814766 0.73 HTR3E (0.46) KCNH2OPRM1OPRL1
SCHEMBL23089139 0.73 HTR3E (0.46) KCNH2OPRM1OPRL1
SCHEMBL17896353 0.71 HTR1A (0.40) HTR1ADRD2DRD4KCNH2CHRNA7
SCHEMBL2609309 0.68 CHRNA7 (0.46) HTR1ADRD2DRD4KCNH2CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021030556-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2021-02-18 WO disclosed