SCHEMBL23009999

SCHEMBL23009999

CC1(C)CCCN1c1nc(Cl)ccc1C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.40
SCN10A Q9Y5Y9 1/20 0.38
CNR2 P34972 1/20 0.36
ACACB O00763 1/20 0.34
PARP2 Q9UGN5 2/20 0.34
TNKS O95271 1/20 0.34
PARP14 Q460N5 1/20 0.34
PARP10 Q53GL7 1/20 0.34
PARP12 Q9H0J9 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
PARP4 Q9UKK3 1/20 0.34
PARP3 Q9Y6F1 1/20 0.34
FFAR2 O15552 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30106504 0.89 KDM5A (0.37) PARP1SCN10ACNR2ACACBFFAR2
SCHEMBL23010272 0.85 PARP1 (0.39) PARP1PARP2TNKSPARP14PARP10
SCHEMBL24773304 0.80 PARP1 (0.36) PARP1ACACBPARP2TNKSPARP14
SCHEMBL21323394 0.78 KIF18A (0.40) SCN10AFFAR2
SCHEMBL28493669 0.77 CFTR (0.37)
SCHEMBL22524695 0.76 FFAR2 (0.34) PARP1ACACBFFAR2
SCHEMBL20998571 0.75 NPC1 (0.46) SCN10A
SCHEMBL21906143 0.74 SCN10A (0.59) SCN10A
SCHEMBL21906101 0.72 SCN10A (0.53) SCN10A
SCHEMBL25629244 0.72 SCN10A (0.33) SCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021030554-A1 PROCESS OF MAKING CFTR MODULATORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2021-02-18 WO disclosed