SCHEMBL23019558

SCHEMBL23019558

COc1cc(NC(=O)NCc2ccccc2)ccc1-c1cnn(C)c1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.61
AAK1 Q2M2I8 1/20 0.60
EP300 Q09472 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.53
AURKB Q96GD4 2/20 0.53
MAPK1 P28482 1/20 0.53
IMPDH2 P12268 3/20 0.50
IMPDH1 P20839 2/20 0.50
TSHR P16473 1/20 0.50
NAMPT P43490 1/20 0.48
ROCK2 O75116 3/20 0.48
ROCK1 Q13464 2/20 0.48
ALDH1A1 P00352 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23019288 0.82 ROCK2 (0.63) RORCEP300AURKBMAPK1TSHR
SCHEMBL19542199 0.77 IDO1 (0.69) RORCAAK1EP300
SCHEMBL3246062 0.77 ROCK2 (0.70) NAMPTROCK2ROCK1ALDH1A1
SCHEMBL20961839 0.77 RORC (1.00) RORC
SCHEMBL29312949 0.76 ROCK2 (0.67) RORCNAMPTROCK2ALDH1A1
SCHEMBL28452637 0.76 RORC (0.87) RORCNAMPT
SCHEMBL28445805 0.75 RORC (0.85) RORCNAMPT
SCHEMBL961096 0.75 AAK1 (0.64) AAK1EP300ALDH1A1
SCHEMBL28454883 0.75 RORC (0.78) RORCAURKBMAPK1TSHR
SCHEMBL5061771 0.74 HTR2A (0.70)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2021-02-24 EP disclosed