SCHEMBL23019288

SCHEMBL23019288

Cn1cc(-c2ccc(NC(=O)NCc3ccccc3)cc2)cn1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.63
ROCK1 Q13464 1/20 0.63
AURKB Q96GD4 2/20 0.61
MAPK1 P28482 1/20 0.61
CLK1 P49759 1/20 0.57
NAMPT P43490 4/20 0.57
RORC P51449 4/20 0.56
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
MAPT P10636 1/20 0.54
TSHR P16473 1/20 0.53
HTT P42858 1/20 0.51
MEN1 O00255 1/20 0.51
TP53 P04637 1/20 0.51
HPGD P15428 1/20 0.51
KMT2A Q03164 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
PTPN1 P18031 1/20 0.51
WNT1 P04628 1/20 0.51
GSK3B P49841 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21426361 0.86 AURKB (0.74) AURKBMAPK1CLK1WNT1GSK3B
SCHEMBL3246062 0.85 ROCK2 (0.70) ROCK2ROCK1CLK1NAMPTMAPT
SCHEMBL18406062 0.83 KIT (0.60) AURKBMAPK1
SCHEMBL21286084 0.82 WNT1 (0.64) NAMPTRORCNPC1RAB9AMAPT
SCHEMBL29312949 0.82 ROCK2 (0.67) ROCK2NAMPTRORCMAPTHTT
SCHEMBL23019558 0.82 RORC (0.61) ROCK2ROCK1AURKBMAPK1NAMPT
SCHEMBL10133206 0.81 ROCK2 (0.80) ROCK2ROCK1NAMPTRORCNPC1
SCHEMBL21426449 0.80 MAPK1 (0.64) AURKBMAPK1CLK1WNT1GSK3B
SCHEMBL23019614 0.79 MAPK1 (0.63) AURKBMAPK1CLK1RORCWNT1
SCHEMBL21426475 0.79 ROCK2 (0.61) ROCK2ROCK1NAMPTRORCNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed
EP-3782986-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2021-02-24 EP disclosed