SCHEMBL29312949

SCHEMBL29312949

COc1ccccc1CNC(=O)Nc1ccc(-c2cnn(C)c2)cc1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.67
MAPT P10636 2/20 0.56
MEN1 O00255 2/20 0.56
HTT P42858 2/20 0.56
KMT2A Q03164 2/20 0.56
HIF1A Q16665 1/20 0.52
NAMPT P43490 4/20 0.51
ALPL P05186 1/20 0.50
RORC P51449 1/20 0.49
ALDH1A1 P00352 2/20 0.49
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
ALOX15 P16050 1/20 0.49
HSD17B10 Q99714 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
CNR1 P21554 1/20 0.48
ANO1 Q5XXA6 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15536148 0.82 AURKB (0.64) MAPTMEN1KMT2ANAMPTALDH1A1
SCHEMBL23019288 0.82 ROCK2 (0.63) ROCK2MAPTMEN1HTTKMT2A
SCHEMBL3243101 0.81 ROCK2 (1.00) ROCK2MAPTMEN1HTTKMT2A
SCHEMBL3246062 0.79 ROCK2 (0.70) ROCK2MAPTMEN1KMT2AHIF1A
SCHEMBL23019558 0.76 RORC (0.61) ROCK2NAMPTRORCALDH1A1
SCHEMBL19349408 0.72 MEN1 (0.53) ROCK2MAPTMEN1KMT2AALDH1A1
SCHEMBL4637492 0.72 KMT2A (0.61) ROCK2MAPTMEN1HTTKMT2A
SCHEMBL20290927 0.70 LRRK2 (0.58) MAPTMEN1KMT2ANAMPT
SCHEMBL20379328 0.70 NAMPT (0.76) MAPTMEN1HTTKMT2ANAMPT
SCHEMBL21286084 0.70 WNT1 (0.64) MAPTMEN1KMT2ANAMPTRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed