SCHEMBL23027463

SCHEMBL23027463

COc1ccc(F)c2c1C(C)(C)CC2

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.35
KDM1A O60341 2/20 0.35
HTR2A P28223 4/20 0.35
HTR2C P28335 4/20 0.35
HTR2B P41595 4/20 0.35
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
ALDH1A1 P00352 3/20 0.33
CYP3A4 P08684 2/20 0.33
MAPT P10636 1/20 0.33
MAOA P21397 1/20 0.33
HPGD P15428 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23027378 0.86 ALDH1A1 (0.36) ADRA1ADRD2DRD3ALDH1A1CYP3A4
SCHEMBL14430374 0.78 ALDH1A1 (0.42) ALDH1A1CYP3A4MAPTHPGDKDM4E
SCHEMBL19870678 0.77 HDAC4 (0.31)
SCHEMBL23027457 0.75 CYP1A2 (0.40) DRD2KDM4EGLA
SCHEMBL9518328 0.75 ADRA1A (0.41) ADRA1AALDH1A1CYP3A4MAOAPTGS1
SCHEMBL14430500 0.71 MAPK1 (0.35) DRD2DRD3GAA
SCHEMBL18053266 0.69 HTR5A (0.46) DRD2DRD3ALDH1A1PTGS1
SCHEMBL31741626 0.68 ADRA1A (0.49) ADRA1AKDM1AHTR2AHTR2CHTR2B
SCHEMBL23027374 0.68 CYP1A2 (0.40) DRD2KDM4EGLA
SCHEMBL10819305 0.67 HDAC4 (0.37) KDM1ADRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021032074-A1 BENZAMIDE FUSED AROMATIC RING DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF IN MEDICINE 江苏恒瑞医药股份有限公司 2021-02-25 WO disclosed