SCHEMBL23049572

SCHEMBL23049572

COC(C)(C)COC(=O)CN

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.31
MGAM O43451 1/20 0.31
GAA P10253 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043538 0.80 ALDH1A1 (0.40) LMNAALDH1A1TSHRTDP1HSD17B10
SCHEMBL1851945 0.79 LMNA (0.34) LMNAKDM4EHSD17B10
Hydrochloric Acid SCHEMBL7314143 0.77 KDM4E (0.35) LMNAKDM4EHSD17B10
SCHEMBL23049725 0.77 LMNA (0.33) LMNAKDM4EHSD17B10
SCHEMBL25383365 0.77 ALDH1A1 (0.39) LMNAALDH1A1TSHRTDP1HSD17B10
SCHEMBL30082486 0.75 KDM4E (0.31) LMNAKDM4E
SCHEMBL19906343 0.75 TET2 (0.32) ALDH1A1TSHRTDP1GAA
SCHEMBL25383367 0.75 ALDH1A1 (0.38) LMNAALDH1A1TSHRTDP1HSD17B10
SCHEMBL9325262 0.74 SERPINE1 (0.32) LMNAKDM4EHSD17B10
SCHEMBL3177457 0.74 CYP1A2 (0.47) LMNAALDH1A1KDM4EHSD17B10MGAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3596064-B1 TOSYLACETATE BASED COMPOUNDS AND DERIVATIVES THEREOF AS PHGDH INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-03-03 EP disclosed