SCHEMBL23058769

SCHEMBL23058769

CCCN(Cc1ccc(F)c(F)c1)C(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
RIPK1 Q13546 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HTT P42858 1/20 0.42
MCHR1 Q99705 1/20 0.41
CYP51A1 Q16850 1/20 0.38
CXCR3 P49682 2/20 0.37
BMP1 P13497 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
BCHE P06276 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
CYP3A4 P08684 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17914544 0.81 MCHR1 (0.52) CYP2D6CYP2C9CYP2C19RIPK1MCHR1
SCHEMBL3971600 0.75 SIGMAR1 (0.52) CYP1A2HTTBCHE
SCHEMBL23058768 0.74 CYP19A1 (0.38) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL17914545 0.73 PYCR1 (0.44) NPSR1HTTMCHR1BCHEHRH3
SCHEMBL23961651 0.73 CYP1A2 (0.43) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL170943 0.73 BCHE (0.51) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL13025108 0.72 PDE2A (0.39) RIPK1HTTHDAC3HDAC6
SCHEMBL23058770 0.72 HDAC3 (0.33) CYP1A2CYP2D6CYP2C9CYP2C19MCHR1
SCHEMBL126441 0.71 TRPA1 (0.46) CYP1A2RIPK1HTT
SCHEMBL20871279 0.71 APLNR (0.49) MCHR1BCHESLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021041588-A1 SUBSTITUTED PYRIDOPYRIMIDINONYL COMPOUNDS USEFUL AS T CELL ACTIVATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-03-04 WO disclosed