SCHEMBL23072050

SCHEMBL23072050

FC(F)(F)c1cnn(-c2ccc(Cl)nn2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
BPTF Q12830 1/20 0.37
ALDH1A1 P00352 2/20 0.36
JUN P05412 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
GABRB3 P28472 2/20 0.35
EPHX2 P34913 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRE P78334 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24240149 0.79 CYP1A2 (0.43) CYP1A2BPTFALDH1A1CHRNB2CHRNA4
SCHEMBL31118756 0.75 EPHX2 (0.40) CYP1A2ALDH1A1NFKB1NFKB2RELA
SCHEMBL11471883 0.73 MAPT (0.48) CYP1A2BPTFALDH1A1KMT2A
SCHEMBL24240163 0.72 EGLN1 (0.41) CYP1A2BPTFALDH1A1KMT2APANK3
SCHEMBL24240164 0.72 BPTF (0.39) CYP1A2BPTFALDH1A1CHRNB2CHRNA4
SCHEMBL30643765 0.72 BPTF (0.39) CYP1A2BPTFALDH1A1CHRNB2CHRNA4
SCHEMBL20075623 0.72 SLC34A1 (0.45) ALDH1A1GABRB3EPHX2GABRPGABRD
SCHEMBL24253730 0.72 GABRB3 (0.38) JUNNFKB1NFKB2RELAGABRB3
SCHEMBL12075244 0.72 EPHX2 (0.45) ALDH1A1GABRB3EPHX2KMT2ASLC34A1
SCHEMBL28606131 0.71 TRPV1 (0.43) JUNNFKB1NFKB2RELAGABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210147393-A1 DIFLUOROMETHYL-PHENYL TRIAZOLES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-05-20 US disclosed
US-10941137-B2 Difluoromethyl-phenyl triazoles BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-03-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10941137-B2 Difluoromethyl-phenyl triazoles GABRA5, GABRB1, GABRA1 CYP1A2 164/4885BPTF 2265/4885ALDH1A1 315/4885
US-20210147393-A1 DIFLUOROMETHYL-PHENYL TRIAZOLES GABRA5, GABRB1, GABRA1 CYP1A2 157/4885BPTF 2248/4885ALDH1A1 308/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.