Bicarbonate

Bicarbonate

SCHEMBL2308797

O=C(O)O.O=C(c1ccc(-c2ccc(Nc3nc4cc(F)ccc4o3)c(F)c2)cc1)C1CCCC1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 5/20 0.49
PIK3CA P42336 1/20 0.43
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41
HDAC6 Q9UBN7 4/20 0.40
HCRTR1 O43613 2/20 0.40
KCNH2 Q12809 2/20 0.39
HCRTR2 O43614 1/20 0.39
CTSL P07711 1/20 0.39
CTSS P25774 1/20 0.39
HPSE Q9Y251 1/20 0.39
CSF1R P07333 1/20 0.38
FAAH O00519 1/20 0.38
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
RAF1 P04049 1/20 0.37
BRAF P15056 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL2314871 0.93 DGAT1 (0.51) DGAT1PIK3CAITGB1ITGA4HDAC6
Bicarbonate SCHEMBL2359226 0.91 DGAT1 (0.42) DGAT1PIK3CAHDAC6KCNH2CSF1R
Bicarbonate SCHEMBL2308864 0.89 DGAT1 (0.41) DGAT1PIK3CAHDAC6KCNH2HPSE
Bicarbonate SCHEMBL2309400 0.89 HDAC6 (0.47) DGAT1PIK3CAHDAC6HCRTR1HCRTR2
SCHEMBL2308795 0.87 DGAT1 (0.65) DGAT1HCRTR1HCRTR2
Bicarbonate SCHEMBL2311135 0.85 DGAT1 (0.44) DGAT1PIK3CAHDAC6CSF1RGAA
Bicarbonate SCHEMBL2308538 0.85 DGAT1 (0.44) DGAT1PIK3CAITGB1ITGA4HCRTR1
Bicarbonate SCHEMBL2314686 0.83 DGAT1 (0.46) DGAT1HDAC6HCRTR1MEN1KMT2A
Bicarbonate SCHEMBL2308696 0.81 CTSL (0.45) DGAT1ITGB1ITGA4HDAC6HCRTR1
SCHEMBL2309693 0.80 DGAT1 (0.67) DGAT1ITGB1ITGA4HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP claimed