SCHEMBL23097447

SCHEMBL23097447

CC(C)c1cc(NS(=O)(=O)c2ccc(Oc3ccc(F)cc3)cc2)c(C(O)O)cc1-c1ccc(COc2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS4 O75173 10/20 0.45
MMP13 P45452 4/20 0.45
ADAMTS5 Q9UNA0 1/20 0.45
ERBB2 P04626 1/20 0.43
ERBB4 Q15303 1/20 0.43
PTGES O14684 1/20 0.42
BCL2L1 Q07817 2/20 0.40
MCL1 Q07820 2/20 0.40
AR P10275 3/20 0.39
MMP2 P08253 1/20 0.39
MMP14 P50281 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
ESR2 Q92731 1/20 0.38
STAT3 P40763 1/20 0.38
CACNA1H O95180 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18152274 0.90 ADAMTS4 (0.47) ADAMTS4MMP13ADAMTS5ERBB2ERBB4
SCHEMBL18151710 0.89 ADAMTS4 (0.45) ADAMTS4MMP13ADAMTS5ERBB2ERBB4
SCHEMBL18151924 0.86 ADAMTS4 (0.49) ADAMTS4MMP13ADAMTS5BCL2L1MCL1
SCHEMBL18152036 0.84 ADAMTS4 (0.48) ADAMTS4MMP13ADAMTS5PTGESBCL2L1
SCHEMBL18174017 0.79 CTSV (0.46) ADAMTS4MMP13ADAMTS5PTGESMCL1
SCHEMBL18152276 0.78 ACLY (0.47) ADAMTS4MMP13ADAMTS5BCL2L1MCL1
SCHEMBL18174100 0.78 PTGES (0.41) ERBB2ERBB4PTGESMAPT
SCHEMBL18151705 0.78 EGFR (0.45) PTGESMCL1MEN1LMNAKMT2A
SCHEMBL18152209 0.78 KDM4E (0.44) ADAMTS4MMP13ADAMTS5ERBB2ERBB4
SCHEMBL18152073 0.77 EGFR (0.44) PTGESMEN1LMNAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3285583-B1 SMALL MOLECULE INHIBITORS OF MCL-1 AND USES THEREOF UNIV MICHIGAN REGENTS (US) 2021-03-17 EP disclosed