SCHEMBL2310172

SCHEMBL2310172

COc1ccc(CC=O)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.44
HTR2A P28223 3/20 0.42
HTR2C P28335 2/20 0.42
ALDH1A1 P00352 3/20 0.42
ERN1 O75460 1/20 0.41
TRIM24 O15164 1/20 0.41
TYR P14679 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
CYP2A6 P11509 1/20 0.39
POLB P06746 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
HSD17B10 Q99714 1/20 0.38
OPRD1 P41143 1/20 0.37
HPGD P15428 2/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
CASP3 P42574 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3928795 0.87 ALDH1A1 (0.41) APLNRHTR2AHTR2CALDH1A1ERN1
SCHEMBL1613798 0.81 APLNR (0.62) APLNRHTR2AHTR2CALDH1A1HSD17B10
SCHEMBL2559819 0.81 HTT (0.45) APLNRALDH1A1ERN1TRIM24TYR
SCHEMBL578049 0.81 ALDH1A1 (0.48) APLNRALDH1A1ERN1TRIM24TYR
SCHEMBL3484107 0.80 APLNR (0.46) APLNRHTR2AHTR2CCYP2A6POLB
SCHEMBL480070 0.80 SLC6A4 (0.43) APLNRHTR2AALDH1A1ERN1TRIM24
SCHEMBL3625530 0.80 POLB (0.57) APLNRALDH1A1ERN1TRIM24TYR
SCHEMBL4006100 0.80 APLNR (0.43) APLNRALDH1A1ERN1TRIM24TYR
SCHEMBL4438609 0.80 CHRM2 (0.47) APLNRALDH1A1ERN1TRIM24TYR
SCHEMBL1134438 0.80 NAAA (0.46) ALDH1A1POLBKDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021150918-A1 4,5,6,7-TETRAHYDROTHIENO[2,3-C]PYRIDINE SUMO INHIBITORS AND USES THEREOF ONCOVALENT THERAPEUTICS INC. (US) 2021-07-29 WO disclosed
EP-2475649-A1 INDENONE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME Korea Research Institute Of Chemical Technology (KR) 2012-07-18 EP disclosed
EP-2348855-A2 SMALL MOLECULE COMPOUNDS FOR STEM CELL DIFFERENTIATION Burnham Institute for Medical Research (US) 2011-08-03 EP disclosed
WO-2011030955-A1 INDENONE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2011-03-17 WO disclosed
WO-2010033643-A2 SMALL MOLECULE COMPOUNDS FOR STEM CELL DIFFERENTIATION BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2010-03-25 WO disclosed