SCHEMBL23102479

SCHEMBL23102479

Cc1c(Br)cccc1-c1nc2c(=O)n(C(=O)OC(C)(C)C)ccc2o1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 1/20 0.36
PIK3CA P42336 1/20 0.36
TP53 P04637 6/20 0.34
TOP2A P11388 2/20 0.34
BUB1 O43683 1/20 0.34
MAPT P10636 5/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
POLB P06746 1/20 0.33
THRB P10828 1/20 0.33
HPGD P15428 3/20 0.32
HSD17B10 Q99714 3/20 0.32
LMNA P02545 3/20 0.32
ALDH1A1 P00352 2/20 0.32
USP2 O75604 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
TSHR P16473 1/20 0.32
NPC1 O15118 2/20 0.32
NFKB1 P19838 2/20 0.32
RAB9A P51151 2/20 0.32
NFKB2 Q00653 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23102420 0.78 TP53 (0.35) TP53TOP2AMAPTSMN1; SMN2HPGD
SCHEMBL23102416 0.78 TP53 (0.31) TP53TOP2AMAPT
SCHEMBL23102583 0.75 USP2 (0.35) TP53TOP2AMAPTSMN1; SMN2HPGD
SCHEMBL23108686 0.74 TOP2A (0.37) TP53TOP2AMAPTSMN1; SMN2HPGD
SCHEMBL23108309 0.73 TNF (0.39) TP53TOP2AMAPTSMN1; SMN2HPGD
SCHEMBL23102593 0.72 SMN1; SMN2 (0.41) TP53TOP2AMAPTSMN1; SMN2HPGD
SCHEMBL23102408 0.72 DUT (0.41) USP2
SCHEMBL23102519 0.71 PIM1 (0.40) PIK3R1PIK3CABUB1PDK4
SCHEMBL19297628 0.69 PIK3R1 (0.44) PIK3R1PIK3CABUB1LMNAL3MBTL1
SCHEMBL23102409 0.68 C1R (0.40) TP53TOP2AMAPTSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021047556-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME AND USE THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed