SCHEMBL23102475

SCHEMBL23102475

O=c1c2cc(Br)oc2ccn1CCO

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.33
PKM P14618 1/20 0.33
P2RX7 Q99572 2/20 0.32
PSMB1 P20618 2/20 0.32
PSMB5 P28074 2/20 0.32
PARP1 P09874 1/20 0.32
GSK3B P49841 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
LMNA P02545 1/20 0.31
ADORA2B P29275 1/20 0.31
PIM1 P11309 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
RECQL P46063 1/20 0.31
TNF P01375 2/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3519282 0.81 PSMB1 (0.32) PSMB1PSMB5PIM1
SCHEMBL23102477 0.76 PDCD1 (0.34) NPSR1PKMALDH1A1RECQL
SCHEMBL1238531 0.75 TNF (0.38) TSHRTNF
SCHEMBL20809182 0.72 PSMB1 (0.41) PSMB1PSMB5ALDH1A1TNF
SCHEMBL1919918 0.72 PSMB1 (0.53) PSMB1PSMB5GSK3BHDAC3HDAC1
SCHEMBL1238094 0.68 CYP1A1 (0.38) PARP1ADORA2BTNF
SCHEMBL13046538 0.67 TNF (0.56) PSMB1PSMB5ALDH1A1LMNATNF
SCHEMBL24184679 0.67 LMNA (0.34) ALDH1A1LMNAADORA2BTNF
SCHEMBL21595152 0.66 HDAC3 (0.39) PARP1ALDH1A1TSHRLMNAADORA2B
SCHEMBL3670650 0.66 L3MBTL1 (0.36) GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021047555-A1 PREPARATION OF AROMATIC HETEROCYCLIC DERIVATIVE AS IMMUNOMODULATOR AND APPLICATION THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed
WO-2021047556-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME AND USE THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed