SCHEMBL2317547

SCHEMBL2317547

Nc1cc(F)c(Cl)cc1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP2A6 P11509 1/20 0.43
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
CSNK2A1 P68400 2/20 0.41
PTGS2 P35354 2/20 0.41
PTGS1 P23219 1/20 0.41
MAP2 P11137 1/20 0.39
FABP4 P15090 2/20 0.39
FABP5 Q01469 1/20 0.37
TSHR P16473 1/20 0.37
MAP4K4 O95819 1/20 0.37
SLC6A4 P31645 1/20 0.36
SMARCA2 P51531 1/20 0.36
SMARCA4 P51532 1/20 0.36
PBRM1 Q86U86 1/20 0.36
FADS1 O60427 1/20 0.36
BACE1 P56817 1/20 0.35
PDE4A P27815 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16119858 0.92 ALDH1A1 (0.43) ALDH1A1HSD17B10CYP2A6ADORA2AADORA1
SCHEMBL21087773 0.84 HSD17B10 (0.50) ALDH1A1HSD17B10PTGS2PTGS1TSHR
SCHEMBL10712308 0.84 ALDH1A1 (0.50) ALDH1A1HSD17B10CYP2A6ADORA1CSNK2A1
SCHEMBL6572708 0.78 GAA (0.52) ALDH1A1HSD17B10CYP2A6ADORA1CSNK2A1
SCHEMBL8734809 0.78 CYP2A6 (0.48) CYP2A6ADORA2AADORA1CSNK2A1PTGS2
SCHEMBL30296558 0.77 CSNK2A1 (0.44) ALDH1A1HSD17B10CYP2A6ADORA2AADORA1
SCHEMBL26456968 0.77 CSNK2A1 (0.44) ALDH1A1HSD17B10CYP2A6ADORA2AADORA1
SCHEMBL2940751 0.77 TDO2 (0.45) ALDH1A1ADORA2AADORA1PTGS2PTGS1
SCHEMBL16615862 0.76 ALDH1A1 (0.62) ALDH1A1HSD17B10CYP2A6ADORA2AADORA1
SCHEMBL17463848 0.74 ALDH1A1 (0.59) ALDH1A1HSD17B10ADORA2AADORA1SMARCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102177137-A 1-phenylpyrrole compounds EXELIXIS INC 2011-09-07 CN disclosed
EP-2349996-A1 1-PHENYLPYRROLE COMPOUNDS Exelixis, Inc. (US) 2011-08-03 EP disclosed
WO-2010042626-A1 1-PHENYLPYRROLE COMPOUNDS EXELIXIS, INC. (US) 2010-04-15 WO disclosed